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DEVELOPMENT OF AN IMPROVED IN VIVO TOOL COMPOUND, VU6001221, FOR NON-COMPETITIVE INHIBITION OF CHT, DISCOVERY AND DEVELOPMENT OF M1 PAMS: BENZOMORPHOLINE AND TETRAHYDROQUINOLINE SERIES, AND DEVELOPMENT OF NOVEL, BRAIN-PENETRANT PAR4 ANTAGONISTS
(2020-06-02)
Here in, we describe the optimization of high-affinity, choline up-take transporter (CHT) antagonist, ML352, to improved in vivo tool compound, VU6001221. VU6001221, a potent and selective CHT inhibitor with significantly ...